{"id":16291,"date":"2020-08-18T03:23:22","date_gmt":"2020-08-18T02:23:22","guid":{"rendered":"http:\/\/blgnoticiassantodomingo.net\/?p=16291"},"modified":"2020-08-18T03:23:24","modified_gmt":"2020-08-18T02:23:24","slug":"descubren-que-un-farmaco-preexistente-para-el-trastorno-bipolar-puede-ser-eficaz-contra-el-coronavirus","status":"publish","type":"post","link":"https:\/\/blgnoticiassantodomingo.net\/index.php\/2020\/08\/18\/descubren-que-un-farmaco-preexistente-para-el-trastorno-bipolar-puede-ser-eficaz-contra-el-coronavirus\/","title":{"rendered":"Descubren que un f\u00e1rmaco preexistente para el trastorno bipolar puede ser eficaz contra el coronavirus"},"content":{"rendered":"\n<h4 class=\"wp-block-heading\">En el marco de su estudio, expertos de EE.UU. evaluaron la mol\u00e9cula de Mpro, enzima clave del SARS-CoV-2 que desempe\u00f1a un papel central en su ciclo de vida.<\/h4>\n\n\n\n<p>Un equipo de cient\u00edficos estadounidenses ha identificado que un f\u00e1rmaco preexistente, utilizado para tratar m\u00faltiples enfermedades, incluidos los trastornos bipolares y la p\u00e9rdida auditiva, podr\u00eda reducir la actividad de una de las debilidades del nuevo coronavirus: su proteasa principal Mpro. Se trata de un avance que puede conducir a una soluci\u00f3n terap\u00e9utica contra el covid-19.<\/p>\n\n\n\n<p>En el marco de su estudio, publicado en la revista&nbsp;<a href=\"https:\/\/advances.sciencemag.org\/content\/early\/2020\/08\/14\/sciadv.abd0345\" target=\"_blank\" rel=\"noreferrer noopener\">Science Advances<\/a>, los expertos de la Universidad de Chicago evaluaron la mol\u00e9cula de Mpro, enzima clave del SARS-CoV-2 que desempe\u00f1a un papel central en su ciclo de vida. Utilizando simulaciones inform\u00e1ticas de \u00faltima generaci\u00f3n, descubrieron que&nbsp;<strong>el f\u00e1rmaco antiinflamatorio ebselen<\/strong>&nbsp;puede ser efectivo en la reducci\u00f3n de su actividad.<\/p>\n\n\n\n<p>\u201cLa proteasa principal es una de las muchas prote\u00ednas del virus que podr\u00edan ser atacadas con medicamentos existentes y reposicionados, y hay miles de compuestos que deben considerarse\u201d,&nbsp;<a href=\"https:\/\/www.eurekalert.org\/pub_releases\/2020-08\/uoc-pds081420.php\" target=\"_blank\" rel=\"noreferrer noopener\">explic\u00f3<\/a>&nbsp;uno de los autores del estudio, Juan de Pablo. \u201cEstamos investigando sistem\u00e1ticamente cada una de las prote\u00ednas involucradas en la funci\u00f3n del virus e investigando sus vulnerabilidades y sus respuestas a una amplia gama de medicamentos\u201d.<\/p>\n\n\n\n<h3 class=\"wp-block-heading\">En busca de debilidades<\/h3>\n\n\n\n<p>Poco despu\u00e9s del brote de covid-19, los cient\u00edficos comenzaron a investigar la estructura del agente causante de la enfermedad, el virus SARS-CoV-2, en busca de debilidades que pudieran verse afectadas por medicamentos nuevos o existentes. Uno de estos objetivos fue la proteasa principal del virus,\u00a0<strong>Mpro<\/strong>. Esta enzima\u00a0<strong>ayuda al pat\u00f3geno a multiplicarse<\/strong>\u00a0dentro de la c\u00e9lula hu\u00e9sped.<\/p>\n\n\n\n<p>Investigaciones anteriores&nbsp;<a href=\"https:\/\/www.nature.com\/articles\/s41586-020-2223-y\" target=\"_blank\" rel=\"noreferrer noopener\">han demostrado<\/a>&nbsp;que varios f\u00e1rmacos disponen de una actividad antiviral prometedora en ensayos basados en c\u00e9lulas, pero el ebselen tiene la inhibici\u00f3n m\u00e1s fuerte de la actividad de Mpro.<\/p>\n\n\n\n<p>Por su parte, investigadores de la Universidad de Chicago, dirigidos por Juan de Pablo, han creado modelos inform\u00e1ticos detallados de la proteasa y el f\u00e1rmaco para comprender exactamente c\u00f3mo podr\u00eda funcionar contra el coronavirus. Result\u00f3 que el&nbsp;<strong>ebselen puede suprimir la actividad de Mpro<\/strong>&nbsp;de dos formas.<\/p>\n\n\n\n<p>En ambos casos, el f\u00e1rmaco interfiere con la inhibici\u00f3n de la actividad de la proteasa, evitando as\u00ed que el coronavirus se multiplique. De esta manera, los resultados de los cient\u00edficos han confirmado que el ebselen es uno de los f\u00e1rmacos prometedores para la lucha contra el covid-19.<\/p>\n\n\n\n<p>Fuente:&nbsp;<strong><a href=\"https:\/\/actualidad.rt.com\/actualidad\/363507-descubren-farmaco-preexistente-trastorno-bipolar\">RT<\/a><\/strong><\/p>\n","protected":false},"excerpt":{"rendered":"<p>En el marco de su estudio, expertos de EE.UU. evaluaron la mol\u00e9cula de Mpro, enzima clave del SARS-CoV-2 que desempe\u00f1a un papel central en su ciclo de vida. Un equipo de cient\u00edficos estadounidenses ha identificado que un f\u00e1rmaco preexistente, utilizado para tratar m\u00faltiples enfermedades, incluidos los trastornos bipolares y la p\u00e9rdida auditiva, podr\u00eda reducir la [&hellip;]<\/p>\n","protected":false},"author":2,"featured_media":16292,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[224],"tags":[1197,3086],"class_list":{"0":"post-16291","1":"post","2":"type-post","3":"status-publish","4":"format-standard","5":"has-post-thumbnail","7":"category-salud","8":"tag-coronavirus","9":"tag-farmaco"},"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v24.9 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Descubren que un f\u00e1rmaco preexistente para el trastorno bipolar puede ser eficaz contra el coronavirus - BLG Noticias<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/blgnoticiassantodomingo.net\/index.php\/2020\/08\/18\/descubren-que-un-farmaco-preexistente-para-el-trastorno-bipolar-puede-ser-eficaz-contra-el-coronavirus\/\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Descubren que un f\u00e1rmaco preexistente para el trastorno bipolar puede ser eficaz contra el coronavirus - BLG Noticias\" \/>\n<meta property=\"og:description\" content=\"En el marco de su estudio, expertos de EE.UU. evaluaron la mol\u00e9cula de Mpro, enzima clave del SARS-CoV-2 que desempe\u00f1a un papel central en su ciclo de vida. 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